Tsuyoshi Saitoh   Mao Amezawa   Jumpei Horiuchi   Yasuyuki Nagumo   Naoshi Yamamoto   Noriki Kutsumura   Ryuichiro Ohshita   Akihisa Tokuda   Yoko Irukayama-Tomobe   Yasuhiro Ogawa   Yukiko Ishikawa   Emi Hasegawa   Takeshi Sakurai   Yasuo Uchida   Tetsu Sato   Hiroaki Gouda   Ryuji Tanimura   Masashi Yanagisawa   Hiroshi Nagase   
European journal of medicinal chemistry 240 114505-114505 2022年10月 [査読有り]
Structurally diverse small compounds are utilized to obtain hit compounds that have suitable pharmacophores in appropriate three-dimensional conformations for the target drug receptors. We have focused on the 1,3,5-trioxazatriquinane skeleton, whi...