Hiroyuki Suzuki   Yuta Kaizuka   Maho Tatsuta   Hiroshi Tanaka   Nana Washiya   Yoshifumi Shirakami   Kazuhiro Ooe   Atsushi Toyoshima   Tadashi Watabe   Takahiro Teramoto   Ichiro Sasaki   Shigeki Watanabe   Noriko S. Ishioka   Jun Hatazawa   Tomoya Uehara   Yasushi Arano   
Journal of Medicinal Chemistry 64(21) 15846-15857 2021年11月 [査読有り]
The high in vivo stability of 2,2-dihydroxymethyl-3-[18F]fluoropropyl-2-nitroimidazole ([18F]DiFA) prompted us to evaluate neopentyl as a scaffold to prepare a radiotheranostic system with radioiodine and astatine. Three DiFA analogues with one, t...